Structure-based drug discovery of a corticotropin-releasing hormone receptor 1 antagonist using an X-ray free-electron laser, Exp Mol Med
Hoyoung Kim, Taehyun Lim, Go Run Ha, Jee-Young Lee, Jun-Woo Kim, Nienping Chang, Si Hyun Kim, Ki Hun Kim,
Jaeick Lee, Yongju Cho, Byeong Wook Kim, Alva Abrahamsson, Sung Hwan Kim, Hyo-Ji Kim, Shan Park, Sang Jae Lee,
Jaehyun Park, Eunhi Cheong, B. Moon Kim, Hyun-Soo Cho*
ArticleA novel therapeutic anti-ErbB3, ISU104 exhibits potent anti-tumorigenic activity by inhibiting
ligand binding and ErbB3 heterodimerizatio, Molecular Cancer Therapeutics
Mirim Hong, Youngki Yoo, Miyoung Kim, Ju Yeon Kim, Jeong Seok Cha, Myung Kyung Choi, Uijin Kim, Kyungyong Kim,
Youngsoo Sohn, Donggoo Bae, Hyun-Soo Cho*, Seoung-Beom Hong* (*co-correspondence)
ArticleComputationally-guided design and affinity improvement of a protein binder targeting a
specific site on HER2, Computational and structural biotechnology journal
Tae Yoon Kim, Jeong Seok Cha, Hoyoung Kim, Yoonjoo Choi, Hyun-Soo Cho*, Hak-Sung Kim* (*co_correspondence)
ArticleDirect binding of TFEα opens DNA binding cleft of RNA polymerase Nature Communications
Sung-Hoon Jun, Jaekyung Hyun, Jeong Seok Cha, Hoyoung Kim, Michael S Bartlett, Hyun-Soo Cho*,
Katsuhiko S Murakami* (*co_correspondence)
ArticleEnzymatic Prenylation and Oxime Ligation for the Synthesis of Stable and Homogeneous
Protein–Drug Conjugates for Targeted Therapy Angewandte Chemie
Joong-jae Lee, Hyo-Jung Choi, Misun Yun, YingJin Kang, Ji-Eun Jung, Yiseul Ryu, Tae Yoon
Kim, Young-je Cha, Hyun-Soo
Cho*, Jung-Joon Min*, Chul-Woong Chung* and
Hak-Sung Kim*,
GC1118, an anti-EGFR antibody with a distinct binding epitope and superior inhibitory activity
against high-affinity EGFR ligands Molecular Cancer Therapeutics
Yangmi Lim, Jiho Yoo, Min-Soo Kim, Minkyu Hur, Eun Hee Lee, Hyung-Suk Hur, Jae-Chul Lee,
Shi-Nai Lee, Tae Wook Park, Kyuhyun
Lee, Ki Hwan Chang, Kuglae Kim, YingJin Kang, Kwang-Won Hong, Se-Ho Kim, Yeon-Gil Kim, Yeup
Yoon, Do-Hyun Nam, Heekyoung
Yang, Dong Geon Kim, Hyun-Soo Cho*, and Jonghwa Won*
Crystal structure and functional characterization of a light-driven chloride
pump having an NTQ motif
Kuglae Kim, Soon-Kyeong Kwon, Sung-Hoon Jun, Jeong Seok Cha, Hoyoung Kim, Weontae Lee, Jihyun F. Kim* and Hyun-Soo Cho*
ArticleStructural basis for arginine glycosylation of host substrates by bacterial effector proteins
Jun Bae Park, Young Hun Kim, Youngki Yoo, Juyeon Kim, Sung-Hoon Jun, Jin Won Cho, Samir El
Qaidi, Samuel Walpole,
Serena Monaco, Ana A. García-García, Miaomiao Wu, Michael P. Hays, Ramon
Hurtado-Guerrero*,
Jesus Angulo*, Philip R. Hardwidge, Jeon-Soo Shin* and Hyun-Soo Cho*